| Cat. No. |
Product Name |
Information |
| PC-27368 |
SRI-9829
NTSR1 agonist
|
SRI-9829 is a potent, selective, nonpeptide full agonist of neurotensin receptor 1 (NTSR1) with EC50 of 0.33 uM, Emax=104%. |
| PC-26998 |
Levocabastine hydrochloride
NTSR2 antagonist
|
Levocabastine hydrochloride (R 50547) is a potent and selective histamine H1-receptor (H1R) antagonist, is also a selective, high affinity neurotensin receptor subtype 2 (NTSR2, NTS2) antagonist with Ki of 17 nM for mNTRS2. |
| PC-26997 |
NTRC-808
NTSR2 agonist
|
NTRC-808 is a potent, selective nonpeptide partial agonist of GPCR neurotensin receptor type 2 (NTS2, NTSR2) with EC50 of 14 nM and Ki of 88 nM, is selective for NTS2 versus NTS1. |