Protease-activated Receptor (PAR) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofProtease-activated Receptor (PAR) Protease-activated Receptor (PAR)

Cat. No.	Product Name	Information
PC-26473	PAR-2 inhibitor I-117 PAR-2 antagonist	PAR-2 inhibitor I-117 is a potent, selective Protease-Activated Receptor-2 (PAR-2) negative allosteric modulator / antagonist with IC50 of 0.09 nM.
PC-23988	SLIGRL-NH2 PAR2 agonist	SLIGRL-NH2 is an agonist of protease-Activated Receptor-2 (PAR-2).
PC-23584	Gestodene PAR1 PAM	Gestodene is a progestogen hormonal contraceptive, also is a positive allosteric modulator of PAR1.
PC-21812	PAR4 antagonist 48 PAR4 antagonist	PAR4 antagonist 48 is a potent and selective quinoxaline-based PAR4 antagonist with IC50 of 1.8 nM in FLIPR calcium mobilization assays, inhibits calcium mobilization in human platelet-rich plasma (PRP) aggregation assay with γ-thrombin with IC50 of 2.1 nM.
PC-20882	PAR2 antagonist C781 PAR2 antagonist	PAR2 antagonist C781 is a potent β-Arrestin biased protease-activated receptor-2 (PAR2) antagonist, effectively reduces 2AT, trypsin and elastase-induced signalling in vitro physiological assays.
PC-20578	TFLLRN-NH2 PAR1 agonist	TFLLRN-NH2 is a potent, PAR1-selective agonist peptide with EC50 of 1.9 uM.
PC-20577	RWJ-58259 PAR1 antagonist	RWJ-58259 (RWJ58259) is a potent, selective thrombin receptor PAR-1 antagonist with binding IC50 of 0.15 uM, and IC50 of 0.07 uM in RASMC calcium mobilization assays.

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