| Cat. No. |
Product Name |
Information |
| PC-20273 |
FR-190997
B2R agonist
|
FR-190997 (FR190997) is a potent, nonpeptide bradykinin (BK) B2 receptor agonist binding IC50 of 1.5 nM (displaced [3H]-BK binding to B2 receptors in guinea-pig ileum membranes). |
| PC-47507 |
Bradykinin
Bradykinin receptor ligand
|
Bradykinin is a 9-amino acid peptide (Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg). |
| PC-45267 |
Icatibant
B2R antagonist
|
Icatibant (HOE 140, JE-049) is a potent, selective and specific antagonist of bradykinin B2 receptor (B2R) with IC50 and Ki of 1.07 nM and 0.798 nM respectively. |
| PC-25718 |
SSR240612
B1R antagonist
|
SSR240612 is a potent, selective, non-peptide antagonist of bradykinin (BK) B(1) receptor, inhibits binding of [(3)H]Lys(0)-des-Arg(9)-BK to B(1) receptor in human fibroblast MRC5 and to recombinant human B(1) receptor expressed in human embryonic kidney cells with Ki of 0.48 and 0.73 nM, respectively. |
| PC-23553 |
R715
B1R antagonist
|
R715 is a potent, selective bradykinin B1 receptor (B1R) antagonist. |