| Cat. No. |
Product Name |
Information |
| PC-43855 |
VX-11e
ERK2 inhibitor
|
VX-11e is a potent, selective, and orally bioavailable inhibitor of ERK2 with Ki of <2 nM. |
| PC-45868 |
SCH772984
ERK1/2 inhibitor
|
SCH772984 is a potent and selective inhibitor of ERK1/ERK2 with IC50 of 4 nM/1 nM, respectively. |
| PC-25096 |
Sonvuterkib
ERK1/2 inhibitor
|
Sonvuterkib (WX001) is a potent, selective ERK1/2 inhibitor. |
| PC-24130 |
SKLB-D18
ERK1/2/5 inhibitor
|
SKLB-D18 is a potent, selective, first-in-class inhibitor of extracellular-regulated kinase 1/2 (ERK1/2) ERK1/2 and ERK5 with IC50 of 38.69/ 40.12 / 59.72 nM respecitvely. |
| PC-22834 |
XMD8-92
ERK5 inhibitor
|
XMD8-92 a specific small-molecule inhibitor of Big mitogen-activated protein kinase 1 (BMK1, ERK5) with Kd of 80 nM, IC50 of 1.5 uM in cell-free assays. |