| Cat. No. |
Product Name |
Information |
| PC-20428 |
ZB-16
GPR119 agonist
|
ZB-16 (ZB40-0016) is a potent, selective GPR119 agonist, increase intracellular cAMP with EC50 of 7.25 nM, stimulates incretin secretion. |
| PC-20426 |
AR231453
GPR119 agonist
|
AR231453 (AR 231453) is the first potent, selective and orally efficacious GPR119 agonist with EC50 of 0.68 nM. |
| PC-72645 |
DA-1241
GPR119 agonist
|
DA-1241 (DA1241) is a novel potent, highly selective GPR119 agonist, activates human GPR119 (EC50=4.37 nM) in increasing cAMP levels in GPR119-overexpressing HEK293 cells. |
| PC-35026 |
AS1269574
GPR119 agonist
|
AS1269574 is a selective, orally available GPR119 agonist with EC50 of 2.5 uM in cell-based cAMP assays. |
| PC-63460 |
MK-8282
GPR119 agonist
|
MK-8282 is a potent, selective, oral GPR119 agonist with EC50 of 10 and 58 nM for hGPR119 and mGPR119, respectively. |
| PC-42879 |
GSK1292263
GPR119 agonist
|
GSK1292263 is a novel potent, selective GPR119 agonist with pEC50 of 6.9 and 6.7 for human and rat GPR119, respectively. |
| PC-60821 |
GSK2041706
GPR119 agonist
|
GSK2041706 is a potent, selective and orally bioavailable GPR119 agonist with EC50 of 4 nM, with good selectivity versus a battery of receptors, ion channels and enzymes. |
| PC-60042 |
Firuglipel
GPR119 agonist
|
Firuglipel (DS8500, DS8500a) is a novel potent, selective, orally available GPR119 agonist with EC50 of 51.5 nM in human GPR119-expressing CHO-K1 cells. |
