Cat. No. |
Product Name |
Information |
PC-72146 |
TAK-041
GPR139 agonist
|
TAK-041 (Zelatriazin, NBI-1065846) is a potent, selective, brain-penetrant GPR139 agonist with EC50 of 22 nM (CHO-T-REx Ca2+ assays), Ki of 119 nM. |
PC-36128 |
GPR139 agonist AC4
GPR139 agonist
|
GPR139 agonist AC4 is a novel small molecule GPR139 receptor agonist with EC50 of 220 nM in calcium mobilization assay in CHO-GPR139 cells. |
PC-45741 |
JNJ-63533054
GPR139 agonist
|
JNJ-63533054 (JNJ63533054) is a potent, selective GPR139 agonist that specifically activates human GPR139 in the calcium mobilization with EC50 of 16 nM. |