c-Kit (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-42449	OSI-930 c-Kit inhibitor	A potent, orally active, dual inhibitor of c-Kit and VEGFR-2 (KDR) with IC50 of 15 nM and 9 nM, respectively.
PC-42455	Masitinib mesylate c-Kit/PDGFR inhibitor	Masitinib (AB-1010) mesylate is a potent tyrosine kinase inhibitor targeting c-Kit and PDGFR with IC50 of 0.15 and 0.05 uM in cell based assays.
PC-42454	Masitinib c-Kit/PDGFR inhibitor	Masitinib (AB1010) is a potent tyrosine kinase inhibitor targeting c-Kit and PDGFR with IC50 of 0.15 and 0.05 uM in cell based assays.
PC-45100	Sitravatinib Multikinase inhibitor	Sitravatinib (MGCD-516) is a broad spectrum small molecule inhibitor that blocks a wide array of RTKs known to be amplified/overexpressed in sarcomas, including c-Kit, PDGFRβ, PDGFRα, c-Met, and Axl (IC50=1.5-30 nM).
PC-42451	Amuvatinib c-Kit inhibitor	Amuvatinib (MP-470) is a potent RTK inhibitor that effectively inhibits c-Kit, PDGFRα and Flt3 with IC50 of 10 nM, 40 nM and 81 nM, respectively.
PC-23095	Labuxtinib c-Kit inhibitor	Labuxtinib is a small molecule inhibitor c-Kit kinase.
PC-21781	BLU-808 c-Kit inhibitor	BLU-808 is a potent and selective wt c-KIT inhibitor, potently inhibits c-KIT–dependent phosphorylation and proliferation with IC50 values in the sub-nanomolar and nanomolar range, respectively.

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