| Cat. No. |
Product Name |
Information |
| PC-61508 |
TAK-259
α1D adrenoceptor antagonist
|
TAK-259 is a potent and selective human α1D adrenoceptor (α1D-AR) antagonist with Ki of 1.1 nM. |
| PC-60734 |
MK-4618
β3 adrenergic receptor agonist
|
MK-4618 (Vibegron, KRP-114V, RVT-901) is a potent and selective full β3 adrenergic receptor agonist with EC50 of 1.1 nM. |
| PC-60704 |
ARC 239 dihydrochloride
α2B adrenoceptor antagonist
|
ARC239 dihydrochloride is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors. |
| PC-60703 |
BRL-44408 maleate
α2A-adrenoceptor antagonist
|
BRL-44408 maleate is a potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors. |
| PC-60702 |
BRL-44408
α2A-adrenoceptor antagonist
|
BRL-44408 is a potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors. |
| PC-70210 |
Levosalbutamol
β2AR agonist
|
Levosalbutamol is a short-acting β2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructive pulmonary disease (COPD). |
| PC-46699 |
Trifluoperazine dihydrochloride
eEF2K inhibitor, α1-adrenergic receptor antagonist
|
Trifluoperazine dihydrochloride is an antiadrenergic, antidopaminergic and anticholinergic agent, potent α1-adrenergic receptor antagonist, also inhibits calcium/calmodulin to eEF2K. |
| PC-45156 |
Dexmedetomidine hydrochloride
α2 adrenoceptor agonist
|
Dexmedetomidine hydrochloride is an agonist of α2-adrenergic receptor with Ki of 1.08 nM. |
| PC-45273 |
Levalbuterol hydrochloride
β2AR agonist
|
Levalbuterol hydrochloride is a short-acting β2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructive pulmonary disease (COPD). |
| PC-45301 |
Metoprolol
β1-adrenoceptor antagonist
|
Metoprolol is a potent, selective and orally active β1-adrenoceptor antagonist, shows anti-inflammation, antitumor and anti-angiogenic properties. |
| PC-45237 |
Guanfacine hydrochloride
α2 adrenoceptor agonist
|
Guanfacine hydrochloride is a selective α2A receptor agonist that can reduce peripheral sympathetic outflow and thus cansues a reduction in peripheral sympathetic tone. |
| PC-43903 |
Olodaterol
β2 adrenoceptor agonist
|
Olodaterol (BI 1744) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2. |
