| Cat. No. |
Product Name |
Information |
| PC-42338 |
Silodosin
α1A-adrenoceptor antagonist
|
Silodosin (KAD3213, KMD3213) is a highly potent, uroselective α1a-adrenoceptor antagonist with Ki of 36 pM. |
| PC-25616 |
Vatinoxan hydrochloride
α2A adrenoceptor antagonist
|
Vatinoxan hydrochloride (MK-467, L-659066) is a potent and selective alpha-2 adrenoceptor (α2A adrenoceptor, α2AR) antagonist with IC50 of 3 nM against the binding of [3H]rauwolscine to rat cerebrocortical membranes, selective over alpha-1 adrenoceptors. |
| PC-25423 |
Formoterol fumarate
β2-adrenoceptor agonist
|
Formoterol fumarate is a potent, selective and long-acting β2-adrenoceptor agonist. |
| PC-25233 |
Imiloxan hydrochloride
α2B adrenoceptor antagonist
|
Imiloxan hydrochloride (RS 21361) is a potent and selective alpha 2B-adrenoceptor antagonist. |
| PC-25232 |
ADRIANA
α2B adrenoceptor antagonist
|
ADRIANA (c545) is a potent, orally active α2B adrenoceptor subtype-specific antagonist with binding Ki of 987 nM, >50-fold selective over α2A adrenoceptor. |
| PC-25231 |
ARC239
α2B adrenoceptor antagonist
|
ARC239 (ARC 239) is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors. |
| PC-24801 |
Salbutamol
β2AR agonist
|
Salbutamol (Albuterol) is a, selective, orally active, short-acting beta-2 adrenergic receptor (β2AR) agonist, 29-fold more selective for beta2 receptors than beta1 receptors. |
| PC-24800 |
BRL-37344
β3AR agonist
|
BRL-37344 (BRL37344) is a potent and selective β3 adrenoceptor (β3AR) agonist with Ki of 287 nM. |
| PC-24799 |
ATR-258
β2AR agonist
|
ATR-258 (Compound 15) is a specific GRK-biased β2 adrenergic receptor (β2AR) agonist with pEC50 of 6.87, increases glucose uptake with low cAMP generation. |
| PC-24569 |
Dabuzalgron
α1A-AR agonist
|
Dabuzalgron (Ro 115-1240) is an orally active and selective α-1A adrenergic receptor agonist with pKi of 7.39 for the displacement of [3H]-prazosin binding to CHO-K1 membranes. |
| PC-24568 |
CCF219B
α1A-AR PAM
|
CCF219B (Compound 3, Cmpd-3) is a potent, selective positive allosteric modulator of the α1A-adrenergic receptor (α1A-AR) with an affinity of 30 nM, 10-50-fold selectivity against the α1B- and α1D-AR subtypes. |
| PC-24491 |
Bisoprolol
β1AR antagonist
|
Bisoprolol is a second-generation, highly selective beta-1 adrenergic receptor (β1AR) antagonist with little activity on β2AR. |
