| Cat. No. |
Product Name |
Information |
| PC-62004 |
Milveterol
β2 adrenoceptor agonist
|
Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold). |
| PC-62003 |
Zinterol hydrochloride
β2 adrenoceptor agonist
|
Zinterol (MJ 9184) is a potent and selective β2 adrenoceptor agonist with pKb of 8.3, displays >2 logs selectivity over β1 (pKb<5.7). |
| PC-62002 |
Zinterol
β2 adrenoceptor agonist
|
Zinterol (MJ 9184) is a potent and selective β2 adrenoceptor agonist with pKb of 8.3, displays >2 logs selectivity over β1 (pKb<5.7). |
| PC-61871 |
PF-00610355
β2 adrenoceptor agonist
|
PF-00610355 (PF 610355) is a potent, selective, and long-acting β2-adrenoreceptor agonist with EC50 of 0.26 nM. |
| PC-61778 |
Xamoterol hemifumarate
β1AR agonist
|
Xamoterol (ICI 118587) is a third-generation adrenergic β1 adrenergic receptor partial agonist that acts as a cardiac stimulant. |
| PC-61776 |
STD-101-D1
β1AR agonist
|
STD-101-D1 is a novel brain permeable, G protein-biased beta-1 adrenergic receptor (ADRB1) partial agonist with EC50 of 16.9 nM. |
| PC-61508 |
TAK-259
α1D adrenoceptor antagonist
|
TAK-259 is a potent and selective human α1D adrenoceptor (α1D-AR) antagonist with Ki of 1.1 nM. |
| PC-60734 |
MK-4618
β3 adrenergic receptor agonist
|
MK-4618 (Vibegron, KRP-114V, RVT-901) is a potent and selective full β3 adrenergic receptor agonist with EC50 of 1.1 nM. |
| PC-60704 |
ARC 239 dihydrochloride
α2B adrenoceptor antagonist
|
ARC 239 dihydrochloride is a potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors. |
| PC-60703 |
BRL-44408 maleate
α2A-adrenoceptor antagonist
|
BRL-44408 maleate is a potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors. |
| PC-60702 |
BRL-44408
α2A-adrenoceptor antagonist
|
BRL-44408 is a potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors. |
| PC-70210 |
Levosalbutamol
β2AR agonist
|
Levosalbutamol is a short-acting β2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructive pulmonary disease (COPD). |
