GPER (GPR30) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofGPER (GPR30) GPER (GPR30)

Cat. No.	Product Name	Information
PC-60270	GPER agonist G-1 GPER agonist	GPER agonist G-1 (Tespria) is potent and selective GPER/GPR30 agonist with Ki of 11 nM, EC50 of 2 nM.
PC-60269	GPER antagonist G36 GPER antagonist	GPER antagonist G36 is a potent, selective, cell-permeable GPER/GPR30 antagonist that inhibits activation by either 17β-estradiol or the GPER-selective agonist G-1 with IC50 of 112 nM and 165 nM, respectively.
PC-60268	G15 GPER antagonist	G-15 (GPR30 inhibitor G15, G15) is a potent, selective GPER/GPR30 antagonist with Ki of 20 nM.
PC-23782	LNS8801 GPER agonist	LNS8801 is a specific, orally available small molecule agonist of G protein–coupled estrogen receptor-1 (GPER), induces both GPER-dependent and GPER-independent effects and elicits potent anticancer activities in vitro and in vivo.

PREV1NEXT