Cat. No. |
Product Name |
Information |
PC-60270 |
GPR30 agonist G-1
GPER agonist
|
GPER/GPR30 agonist G-1 (Tespria) is potent and selective GPER/GPR30 agonist with Ki of 11 nM, EC50 of 2 nM. |
PC-60269 |
GPER antagonist G36
GPER antagonist
|
GPER antagonist G36 is a potent, selective, cell-permeable GPER/GPR30 antagonist that inhibits activation by either 17β-estradiol or the GPER-selective agonist G-1 with IC50 of 112 nM and 165 nM, respectively. |
PC-60268 |
G15
GPER antagonist
|
G-15 (GPR30 inhibitor G15, G15) is a potent, selective GPER/GPR30 antagonist with Ki of 20 nM. |