| Cat. No. |
Product Name |
Information |
| PC-43317 |
MK-0354
GPR109A agonist
|
MK-0354 is a potent, selective niacin receptor GPR109A partial agonist with EC50 of 1.65 and 1.08 uM for hGPR109A and mGPR109A in the whole cell cAMP assays. |
| PC-42694 |
MK-6892
GPR109A agonist
|
MK-6892 is a potent and selective high affinity niacin receptor (GPR109A) full agonist with Ki of 4.0 nM, EC50 of 16 nM in GTPγS assay. |
| PC-21439 |
GSK256073
GPR109A agonist
|
GSK256073 is a highly potent, selective agonist of hydroxy-carboxylic acid receptor 2 (HCA2, HM74A/GPR109A) with pEC50 of 7.5, 100-fold selective over HCA3 (pEC50=5.6). |
| PC-21427 |
MK-1903
GPR109A agonist
|
MK-1903 is potent and selective agonist of GPR109a with EC50 of 12.9 nM, Emax 102%. |
| PC-21426 |
SCH900271
GPR109A agonist
|
SCH900271 is a potent nicotinic acid receptor GPR109A agonist with EC50 of 2 nM in hu-GPR109a assays. |
