| Cat. No. |
Product Name |
Information |
| PC-42234 |
SNAP 37889
GalR3 antagonist
|
SNAP 37889 (HT-2157) is a potent, selective galanin-3 receptor (GalR3) antagonist with Ki of 17.44 nM, displays highly selective for Gal3 over the Gal1 and Gal2 subtypes (both Ki >10 uM). |
| PC-23341 |
SNAP 398299
GALR3 antagonist
|
SNAP 398299 a highly water-soluble analog of SNAP 37889 and selective, high-affinity antagonist of Gal3 receptor (GALR3) with Ki of 5.33 nM, no significant affinity for Gal1 and Gal2 receptors (Ki>1000 nM). |
| PC-23339 |
M617
GALR1 agonist
|
M617 is a potent, selective galanin receptor 1 (GALR1) agonist with Ki values of 0.23 nM and 5.71 nM for GALR1 and GALR2, respectively |
| PC-23338 |
M871
GALR2 antagonist
|
M871 (Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide) is a potent, selective galanin receptor type 2 (GALR2) antagonist with Ki value of 13.1 nM, >30-fold selective over GALR2. |
| PC-23337 |
Spexin
GALR2/3 ligand
|
Spexin (SPX) is a pleiotropic peptide with highly conserved protein sequence and ligand of GalR2/GalR3 receptors. |
| PC-23336 |
M1145
GALR2 agonist
|
M1145 is a chimeric peptide, potent, selective galanin receptor type 2 (GALR2) agonist with Ki of 6.55 nM, >50-fold selective over GALR1 (Ki=587 nM) and GALR3 (Ki=497 nM). |
