| Cat. No. |
Product Name |
Information |
| PC-38133 |
UCSF7447
MT-1 inverse agonist
|
UCSF7447 (UCSF-7447, ZINC555417447) is a potent, selecive, brain permeable melatonin receptor MT-1 inverse agonist with Ki of 304 nM (hMT-1). |
| PC-61335 |
Piromelatine
Melatonin receptor/5-HT agonist
|
Piromelatine (Neu-P11) is a melatonin melatonin receptor MT1/MT2 and serotonin 5-HT1A/5-HT1D receptor agonist. |
| PC-45162 |
Agomelatine L( )-Tartaric acid
|
A melatonin receptor agonist of MT1 (Ki=0.1nM) and MT2 (Ki=0.12nM), and a 5-HT2C (Ki=631nM) receptor antagonist. |
| PC-45161 |
Agomelatine hydrochloride
Melatonin receptor agonist
|
Agomelatine hydrochloride (S-20098) melatonin receptor agonist of MT1 (Ki=0.1nM) and MT2 (Ki=0.12nM), and a 5-HT2C (Ki=631nM) receptor antagonist. |
| PC-45160 |
Agomelatine
Melatonin receptor agonist
|
Agomelatine (S-20098) is a melatonin receptor agonist of MT1 (Ki=0.1nM) and MT2 (Ki=0.12nM), and a 5-HT2C (Ki=631nM) receptor antagonist. |
| PC-23432 |
Prazosin
MT3 receptor antagonist
|
Prazosin is an α-adrenergic receptor antagonist, and selective MT3 melatonin receptor antagonist. |
| PC-23431 |
MT2 antagonist DH97
MT2 receptor antagonist
|
DH97 is a potent and selective antagonist of MT2 melatonin receptor with pKi value of 8.03 for human MT2 receptor, shows 89- and 229-fold selectivity over human MT1 and Xenopus mel1c receptor subtypes. |
| PC-23430 |
Luzindole
Melatonin receptor antagonist
|
Luzindole (N-0774) is a potent, selective melatonin receptor antagonist with Ki of 10.2 nM and 158 nM for human MT2 and MT1, respectively. |
