Cat. No. |
Product Name |
Information |
PC-42779 |
GW843682X
PLK1/3 inhibitor
|
GW843682X is a potent and selective inhibitor of PLK1 (IC5=2.2 nM) and PLK3 (IC50=9 nM). |
PC-23368 |
TC-S 7005
PLK2 inhibitor
|
TC-S 7005 is a potent, selective polo-like kinase 2 (PLK2) inhibitor with IC50 of 4 nM, 24 nM and 214 nM for PLK2, PLK3, and PLK1, respectively. |
PC-22312 |
NMS-P937
PLK1 inhibitor
|
NMS-P937 (Onvansertib, NMS-1286937) is a potent, selective and orally available PLK1 inhibitor with IC50 of 2 nM. |
PC-21170 |
SBE13
PLK1 inhibitor
|
PLK1 inhibitor SBE13 is a potent, selective PLK1 inhibitor with IC50 of 0.2 nM, with little to no inhibition against PLK2/PLK3 (IC50, 65 uM/875 nM). |
PC-21169 |
Ro3280
PLK1 inhibitor
|
Ro3280 is a potent, specific PLK1 inhibitor with IC50/Kd of 3/0.09 nM, respectively, shows no activity against PLK2/3. |