Cat. No. |
Product Name |
Information |
PC-45677 |
LJH-685
RSK inhibitor
|
LJH-685 is a potent and specific pan-RSK inhibitor with IC50s of 6 nM,5 nM and 4 nM for RSK1,RSK2 and RSK3 respectively. |
PC-45919 |
CMK
RSK2 inhibitor
|
CMK is an irreversible inhibitor of the CTD of RSK2 with similar potency as Fmk, also potently inhibits a Fyn mutant in which Val285 was replaced with Cys (IC50=1 nM). |
PC-45920 |
FMK
RSK inhibitor
|
FMK is an irreversible inhibitor of the CTD of RSK1 and RSK2 with IC50 of 15 nM for wt RSK2. |
PC-42627 |
BI-D1870
RSK inhibitor
|
BI-D1870 is a potent, specific ATP-competitive inhibitor of RSK isoforms with IC50 of 10-30 nM for RSK1/2/3/4. |