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Cat. No. Product Name Information
PC-35949

SR146131

CCK1 inhibitor

SR146131 (SR-146131) a small molecule positive allosteric modulator of the type 1 cholecystokinin receptor (CCK1R) with pEC50 of 10.34.
PC-70239

L-365260

CCK2 inhibitor

L-365260 (L365260) is a potent, selective, orally active cholecystokinin receptor 2 (CCK2) antagonist with IC50 of 2 nM.
PC-70198

PF-04756956

CCK1 inhibitor

PF-04756956 is a potent, selective CCK1 receptor agonist with EC50 of 0.47 nM.
PC-70197

CE-326597

CCK1 agonist

CE-326597 is a potent, selective agonist of the human and rat CCK1 receptor with Ki of 36 nM.
PC-70196

JNJ-26070109

CCK2 inhibitor

JNJ-26070109 is a novel, potent, selective orally active CCK-2 receptor antagonist with pKi of 8.49 for hCCK2.
PC-60082

Netazepide

CCK2 inhibitor

Netazepide (YF476, Sograzepide) is a potent, selective and orally active gastrin/CCK-2 antagonist with IC50 of 0.1 nM.
PC-60036

Ceclazepide

CCK2 inhibitor

Ceclazepide is a potent, selective cholecystokinin receptor CCK2 antagonist for treatment of gastroesophageal reflux disease (GERD).
PC-45389

Z-360

CCK2 inhibitor

Z-360 (Nastorazepide) is a novel potent, orally active CCK-2/gastrin receptor antagonist with Ki of 0.47 nM.
PC-22021

Devazepide

CCK1 inhibitor

Devazepide (L-364,718) is a potent, competitive, selective and orally active nonpeptide antagonist of peripheral cholecystokinin (CCK) receptor with IC50 of 81 pM, 45 pM and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors.
PC-22020

A71623

CCK1 agonist

A-71623 (A71623) is a cholecystokinin tetrapeptide (30-33) analogue as potent, highly selective CCK-A (CCK1) cholecystokinin receptor agonist with binding IC50 of 3.7 nM, >1000-fold selective over CCK-B receptor.
PC-22019

GW-5823

CCK1 agonist

GW5823 (GW-5823) a potent, selective orally active, gut-selective CCK1 receptor (CCK-A receptor) agonist with binding pIC50 of 7.64, ED50 of 109 nM in functional  assays.

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