| Cat. No. |
Product Name |
Information |
| PC-72645 |
DA-1241
GPR119 agonist
|
DA-1241 (DA1241) is a novel potent, highly selective GPR119 agonist, activates human GPR119 (EC50=4.37 nM) in increasing cAMP levels in GPR119-overexpressing HEK293 cells. |
| PC-35026 |
AS-1269574
|
AS-1269574 is a selective, orally available GPR119 agonist with EC50 of 2.5 uM in cell-based cAMP assays. |
| PC-60042 |
Firuglipel
|
Firuglipel (DS-8500, DS8500a) is a novel potent, selective, orally available GPR119 agonist with EC50 of 51.5 nM in human GPR119-expressing CHO-K1 cells, displays no significant effect on 66 receptors, channels, or transporters. |
| PC-20444 |
PSN632408
GPR119 agonist
|
PSN632408 (PSN 632408) is a selective small-molecule GPR119 agonist with cAMP EC50 of 7.9 and 5.6 uM for mouse and human GPR119 receptor, respectively. |
| PC-20443 |
GPR119 agonist 27
GPR119 agonist
|
GPR119 agonist 27 is a potent, selective and orally bioavailable GPR119 agonist with EC50 of 4.6 nM (hGPR119). |
| PC-20442 |
JTP-109192
GPR119 agonist
|
JTP-109192 (JTP109192) is a potent GPR119 agonist with EC50 of 3.6. 4.5 and 5.2 nM for human, rat and mouse GPR119 respectively (increased intracellular cAMP levels). |
| PC-20440 |
AS1907417
GPR119 agonist
|
AS1907417 is a potent, selective GPR119 agonist with cAMP EC50 of 1.1 uM (human GPR119). |
| PC-20439 |
AS1535907
GPR119 agonist
|
AS1535907 is a potent GPR119 agonist with EC50 of 4.8 uM in HEK293 cells stably expressing human GPR119. |
| PC-20437 |
APD668
GPR119 agonist
|
APD668 (JNJ-28630368) is a potent and selective GPR119 agonist with EC50 of 2.7 and 33 nM for huamn and rat GPR119, respectively. |
| PC-20436 |
BMS-986034
GPR119 agonist
|
BMS-986034 (BMS 986034) is a potent and selective GPR119 agonist. |
| PC-20435 |
BMS-903452
GPR119 agonist
|
BMS-903452 (BMS 903452) is a potent and selective GPR119 agonist with EC50 of 14 nM. |
| PC-20432 |
MBX-2982
GPR119 agonist
|
MBX-2982 (SAR 260093) is a potent, selective, orally-available GPR119 agonist with pEC50 of 8.33 in GPR119 cAMP assays. |
