| Cat. No. |
Product Name |
Information |
| PC-23321 |
Pranlukast
CysLT antagonist
|
Pranlukast (SB 205312, ONO-1078) is a highly potent, selective and competitive leukotriene antagonist, inhibits [3H]LTE4, [3H]LTD4, and [3H]LTC4 bindings to lung membranes with Ki values of 0.63 nM, 0.99 nM, and 5640 nM, respectively. |
| PC-23320 |
Montelukast sodium
CysLT1 antagonist
|
Montelukast (MK0476) sodium is a potent, selective and orally active antagonist of cysteinyl leukotriene receptor 1 (CysLT1) with Ki of 0.18 nM, 4 nM and 0.52 nM in guinea pig lung, sheep lung and U937 cell plasma membrane preparations respectively. |
| PC-23319 |
Montelukast
CysLT1 antagonist
|
Montelukast (MK0476) is a potent, selective and orally active antagonist of cysteinyl leukotriene receptor 1 (CysLT1) with Ki of 0.18 nM, 4 nM and 0.52 nM in guinea pig lung, sheep lung and U937 cell plasma membrane preparations respectively. |
| PC-21589 |
LY255283
BLT2 inhibitor
|
LY255283 is a selective, competitive antagonist of leukotriene B4 receptor (BLT2) with IC50 of 1 uM, 10-fold selective over BLT1 receptor. |
| PC-21194 |
U75302
LTB4 receptor 1 inhibitor
|
U75302 is a specific leukotriene B4 receptor 1 (LTB4 receptor 1, BLTR1, BLT1) inhibitor, effectively block LTB4 responses. |
