| Cat. No. |
Product Name |
Information |
| PC-72913 |
BAY-298
LH-R inhibitor
|
BAY-298 (BAY298) is a highly potent, selective luteinizing hormone receptor (LH-R) inhibitor with IC50 of 96 nM and 23 nM for hLH-R and rLH-R, respectively. |
| PC-72912 |
BAY-899
LH-R inhibitor
|
BAY-899 (BAY899) is a highly potent, selective luteinizing hormone receptor (LH-R) inhibitor with IC50 of 185 nM and 46 nM for hLH-R and rLH-R, respectively. |
| PC-43101 |
Triptorelin
LHR agonist
|
Triptorelin is a synthetic decapeptide agonist analog of luteinizing hormone releasing hormone (LHRH), shows greater potency than endogenous LHRH, triptorelin reversibly represses gonadotropin secretion.. |
| PC-62756 |
Org 42599 free base
LHR agonist
|
Org 42599 is a cell-permeant, allosterically binding, small-molecule agonist of luteinizing hormone (LH) receptor that rescues the folding and cell surface expression mutant mutant human LH receptors A593P and S616Y (EC50=70.8 nM). |
| PC-62038 |
Org 42599
LHR agonist
|
Org 42599 is a cell-permeant, allosterically binding, small-molecule agonist of luteinizing hormone (LH) receptor that rescues the folding and cell surface expression mutant mutant human LH receptors A593P and S616Y (EC50=70.8 nM). |
| PC-42085 |
Sufugolix
LHRH receptor antagonist
|
Sufugolix (TAK-013) is a highly potent and orally bioavailable non-peptide antagonist of luteinizing hormone-releasing hormone (LHRH) receptor with binding and functional IC50 of 0.1 and 0.06 nM for human LHRH, respectively. |
