Cat. No. |
Product Name |
Information |
PC-61118 |
BMS-814580
MCHR1 inhibitor
|
BMS-814580 is a highly potent, subtype-selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 17 nM, without inhibitory activity for MCHR2 at 10 uM. |
PC-22854 |
KRX-104130
MCHR1 antagonist
|
KRX-104130 is a potent melanin-concentrating hormone receptor 1 (MCHR1) antagonist with IC50 of 0.02 uM, shows no cardiotoxicity. |
PC-22723 |
MCHR2 antagonist 38
MCHR2 antagonist
|
MCHR2 antagonist 38 is a potent and specific MCH receptor subtype 2 (MCHR2) antagonist with IC50 of 1 nM in MCHR2 Ca+2 FLIPR assay, Ki of 13 nM. |
PC-61119 |
BMS 814580 phosphate
|
A highly potent, subtype-selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 17 nM, without inhibitory activity for MCHR2 at 10 uM. |