| Cat. No. |
Product Name |
Information |
| PC-61532 |
NGD-4715
MCHR1 inhibitor
|
NGD-4715 is a potent, selective, non-peptide antagonist of MCHR1 (Melanin-concentrating hormone receptor 1), has anxiolytic, antidepressant and anorectic effects. |
| PC-61531 |
ALB-127158
MCHR1 inhibitor
|
ALB-127158 is a potent (IC50=7 nM), selective, non-peptide antagonist of MCHR1 (Melanin-concentrating hormone receptor 1) for treatment of obesity.. |
| PC-61530 |
AMG-076
MCHR1 inhibitor
|
AMG-076 is a potent, selective, non-peptide antagonist of MCHR1 (Melanin-concentrating hormone receptor 1) with binding IC50 of 0.6 nM, with dramatically reduced hERG liability (IC50>5 uM). |
| PC-61529 |
T-226296
MCHR1 inhibitor
|
T-226296 is a potent, selective, non-peptide antagonist of MCHR1 (Melanin-concentrating hormone receptor 1) with IC50 of 5.5 nM and 8.6 nM for human and rat MCHR1, respectively. |
| PC-61528 |
SNAP-7941
MCHR1 inhibitor
|
SNAP-7941 is a selective, high-affinity, and competitive MCH1 receptor (MCHR1) antagonist with Ki of 15 nM. |
| PC-61527 |
SNAP-94847
MCHR1 inhibitor
|
SNAP-94847 is a selective, high-affinity, and competitive MCH1 receptor (MCHR1) antagonist with Ki of 1.69 nM. |
| PC-61526 |
SNAP-94847 hydrochloride
MCHR1 inhibitor
|
SNAP-94847 hydrochloride is a selective, high-affinity, and competitive MCH1 receptor (MCHR1) antagonist with Ki of 1.69 nM. |
| PC-61512 |
BI 186908
MCHR1 inhibitor
|
BI 186908 is a potent and selective MCH1 receptor (MCHR1) antagonist with IC50 of 22 nM, Ki of 14 nM. |
| PC-61510 |
AZD1979
MCHR1 inhibitor
|
AZD1979 is a potent, selective melanin concentrating hormone receptor 1 (MCH-R1, MCHR1) antagonist with binding Ki of 12.2 nM. |
| PC-61122 |
BMS-830216
MCHR1 inhibitor
|
The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM. |
| PC-61121 |
BMS-819881
MCHR1 inhibitor
|
A potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM. |
| PC-61120 |
GW803430
MCHR1 inhibitor
|
GW803430 is a potent, specific, orally active melanin concentrating hormone receptor 1 (MCHR1) inhibitor with kI of 3.8 nM, >100-fold selectivity over a battery of GPCRs, ion channels and enzymes. |
