Pyruvate Dehydrogenase Kinase (PDK) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofPyruvate Dehydrogenase Kinase (PDK) Pyruvate Dehydrogenase Kinase (PDK)

Cat. No.	Product Name	Information
PC-21872	M77976 PDK4 inhibitor	M77976 is a selective inhibitor of pyruvate dehydrogenase kinase 4 (PDK4) with IC50 of 648 uM, binds to the ATP-binding pocket of PDK4.
PC-63500	PS10 PDK inhibitor	PS10 (PDK inhibitor PS10) is a novel potent and highly selective pyruvate dehydrogenase kinase (PDK) inhibitor with IC50 values of 0.8 μM, 0.76 μM, 2.1 μM and 21.3 μM for PDK2, PDK4, PDK1, and PDK3, respectively.
PC-23745	Radicicol PDK1/PDK3 inhibitor	Radicicol is an inhibitor of Hsp90 with IC50 value <1 μM, also inhibits pyruvate dehydrogenase kinase (PDHK, PDK) with IC50 of 230 μM (PDK1) and 400 μM (PDK3).
PC-23744	AZD7545 PDHK inhibitor	AZD7545 is a potent, selective inhibitor of pyruvate dehydrogenase kinase (PDHK, PDK) with IC50 of 36.8 nM and 6.4 nM for PDHK1 and PDHK2 respectively.
PC-23723	Sodium dichloroacetate PDK1 inhibitor	Sodium dichloroacetate is a small molecule inhibitor of pyruvate dehydrogenase kinase 1 (PDK1, PDHK1), decreases lactic acid in the tumor microenvironment.

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