| Cat. No. |
Product Name |
Information |
| PC-49080 |
J-2156
SST4 agonist
|
J-2156 is a highly potent, selective somatostatin SST4 receptor agonist with binding Ki value of 1.2 nM (hSST4R), >400-fold selectivity over other human somatostatin receptor subtypes. |
| PC-38746 |
CRN02481
SST5 agonist
|
CRN02481 is a potent and selective SST5 receptor agonist with EC50 of 0.37 nM (human SST5), with excellent selectivity against SST1, SST2, SST3 and SST4 receptors. |
| PC-38007 |
Paltusotine
SST2 agonist
|
Paltusotine (CRN00808) is an orally bioavailable, nonpeptide, somatostatin receptor subtype 2 (SST2) agonist with EC50 of 0.25 nM. |
| PC-61088 |
MK-4256
SSTR3 antagonist
|
MK-4256 is a potent, selective, orally active somatostatin receptor SSTR3 antagonist with binding Ki of 0.66 nM, >500-fold selectivity over SSTR1/2/4/5. |
| PC-61087 |
MK-1421
SSTR3 antagonist
|
MK-1421 is a potent, selective, orally active somatostatin receptor SSTR3 antagonist with binding Ki of 2.3 nM, >2,500-fold selectivity over SSTR1/2/4/5 (IC50>5 uM). |
| PC-45184 |
Octreotide acetate
SSTR agonist
|
Octreotide (SMS 201-995) acetate is an octapeptide that mimics natural somatostatin pharmacologically, that is 200 times more potent than somatostatin. |
| PC-46000 |
Pasireotide L-aspartate salt
SSTR agonist
|
Pasireotide (SOM230) L-aspartate is a potent, stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (pKi=8.2/9.0/9.1/<7.0/9.9 for sst1/2/3/4/5, respectively). |
| PC-45999 |
Pasireotide ditrifluoroacetate
SSTR agonist
|
Pasireotide ditrifluoroacetate (SOM230) is a potent, stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (pKi=8.2/9.0/9.1/<7.0/9.9 for sst1/2/3/4/5, respectively). |
| PC-44950 |
Pasireotide
SSTR agonist
|
A potent, stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (pKi=8.2/9.0/9.1/<7.0/9.9 for sst1/2/3/4/5, respectively). |
| PC-23186 |
L-054,264
SST2 agonist
|
L-054,264 is a potent, selective non-peptide human somatostatin receptor subtype 2 (sst2) agonist with Ki of 1.6 nM, >1000-fold selective over other somatostatin receptor subtypes. |
| PC-22364 |
Octreotide
SSTR agonist
|
Octreotide (SMS 201-995) is an octapeptide that mimics natural somatostatin pharmacologically, that is 200 times more potent than somatostatin. |
| PC-22363 |
Pasireotide acetate
SSTR agonist
|
Pasireotide (SOM230) acetate is a potent, stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (pKi=8.2/9.0/9.1/<7.0/9.9 for sst1/2/3/4/5, respectively). |
