| Cat. No. |
Product Name |
Information |
| PC-42121 |
A-922500
DGAT-1 inhibitor
|
A-922500 (A922500) is a potent, selective and orally bioavailable DGAT-1 inhibitor with IC50 of 9 and 22 nM against human and mouse DGAT-1, respectively. |
| PC-45795 |
T863
DGAT1 inhibitor
|
T-863 is a potent and selective, cell-permeable DGAT1 inhibitor that binds to the oleoyl-CoA binding pocket of DGAT1 with IC50 of 17 nM in TLC assay. |
| PC-21285 |
PF-07202954
DGAT2 inhibitor
|
PF-07202954 is a potent, selective next-generation DGAT2 inhibitor with IC50 of 10 nM (hDGAT2). |
| PC-21222 |
TP-020
MGAT2 inhibitor
|
TP-020 is a potent, selective, orally active inhibitor of monoacylglycerol acyltransferase (MGAT2) with IC50 of 7.8 and 2.4 nM for human and mouse MGAT2, respectively. |
| PC-21221 |
BMS-986172
MGAT2 inhibitor
|
BMS-986172 is a highly potent, selective monoacylglycerol acyltransferase 2 (MGAT2) inhibitor with IC50 of 4.6 nM (human MGAT2). |
| PC-62952 |
JTT-553 benzosulfonate
|
JTT-553 is a novel potent, selective DGAT-1 inhibitor with IC50 of 2.38 nM, shows no inhibitory activity for human DGAT2 and ACA T1 (IC50>10 uM). |
