| Cat. No. |
Product Name |
Information |
| PC-24954 |
Fosrolapitant
NK1R antagonist
|
Fosrolapitant is a potent, selective neurokinin-1 receptor (NK1R) antagonist. |
| PC-24029 |
WIN 62577
NK1 receptor antagonist
|
WIN 62577 (WIN 62,577) is a selective antagonist of tachykinin NK1 receptor, also is an allosteric enhancer with micromolar potency at muscarinic M3 receptor, also is a highly efficacious inhibitor of main protease (Mpro) of SARS-CoV-2. |
| PC-23421 |
EB1002
NK2R agonist
|
EB1002 is a potent, selective, long-acting neurokinin 2 receptor (NK2R), enhances insulin sensitization. |
| PC-23398 |
Vofopitant dihydrochloride
NK1 receptor antagonist
|
Vofopitant dihydrochloride (GR 205171A) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist, inhibits [3H]SP binding to the NK1 receptor with pKi values of 9.5 and 10.6 in rat and human membranes respectively. |
| PC-23397 |
Vofopitant
NK1 receptor antagonist
|
Vofopitant (GR205171) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist, inhibits [3H]SP binding to the NK1 receptor with pKi values of 9.5 and 10.6 in rat and human membranes respectively. |
| PC-22655 |
SR140333B
NK1 receptor antagonist
|
Nolpitantium besilate (SR140333B) is a potent, selective, non-peptide NK1 receptor antagonist with Ki of 0.74 nM, IC50 of 1.6 nM. |