Cat. No. |
Product Name |
Information |
PC-23397 |
Vofopitant
NK1 receptor antagonist
|
Vofopitant (GR205171) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist, inhibits [3H]SP binding to the NK1 receptor with pKi values of 9.5 and 10.6 in rat and human membranes respectively. |
PC-22655 |
SR140333B
NK1 receptor antagonist
|
Nolpitantium besilate (SR140333B) is a potent, selective, non-peptide NK1 receptor antagonist with Ki of 0.74 nM, IC50 of 1.6 nM. |
PC-21757 |
Elinzanetant
NK1/3R inhibitor
|
Elizanetant (NT-814) is an orally active, selective neurokinin (NK) receptors 1 and 3 antagonist, modulates reproductive hormone secretion. |