| Cat. No. |
Product Name |
Information |
| PC-27026 |
Fosnetupitant chloride monohydrochloride
NK1R antagonist
|
Fosnetupitant chloride monohydrochloride is a phosphorylated prodrug formulation of netupitant and selective neurokinin-1 receptor (NK1R) antagonist with pKi of 9.5, >1000-fold selective over NK3R. |
| PC-27025 |
Fosnetupitant
NK1R antagonist
|
Fosnetupitant is a phosphorylated prodrug formulation of netupitant and selective neurokinin-1 receptor (NK1R) antagonist with pKi of 9.5, >1000-fold selective over NK3R. |
| PC-25517 |
Fosaprepitant dimeglumine
NK1R antagonist
|
Fosaprepitant dimeglumine (MK-0517) is a prodrug of Aprepitant (PC-42185), which is a potent, selective neurokinin-1 receptor (NK1R)antagonist |
| PC-25117 |
CP-99994 dihydrochloride
NK1 antagonist
|
CP-99994 dihydrochloride is a selective, high-affinity Neurokinin-1 (substance P) receptor (NK1R) antagonist with binding Ki of 0.17 nM. |
| PC-25041 |
Dazodeunetant
NK3R antagonist
|
Dazodeunetant is a potent, selective neurokinin 3 receptor (NK3R) antagonist. |
| PC-24954 |
Fosrolapitant
NK1R antagonist
|
Fosrolapitant is a potent, selective neurokinin-1 receptor (NK1R) antagonist. |
| PC-24029 |
WIN 62577
NK1 receptor antagonist
|
WIN 62577 (WIN 62,577) is a selective antagonist of tachykinin NK1 receptor, also is an allosteric enhancer with micromolar potency at muscarinic M3 receptor, also is a highly efficacious inhibitor of main protease (Mpro) of SARS-CoV-2. |
| PC-22655 |
SR140333B
NK1 receptor antagonist
|
Nolpitantium besilate (SR140333B) is a potent, selective, non-peptide NK1 receptor antagonist with Ki of 0.74 nM, IC50 of 1.6 nM. |
