Cat. No. |
Product Name |
Information |
PC-70191 |
Ibodutant
|
A potent and selective linear tachykinin NK2 receptor antagonist with pKb of 9.3. |
PC-70190 |
RP-67580
|
A potent and selective tachykinin NK1 receptor antagonist with Ki of 2.9 nM. |
PC-70189 |
Saredutant
|
A potent and selective non-peptide antagonist of the neurokinin A (NK2) receptor. |
PC-60173 |
NK1-IN-9
|
A potent, orally active, dual NK1 receptor antagonist (IC50=0.5 nM) and SERT inhibitor (IC50=5.2 nM). |
PC-42191 |
Maropitant
|
A selective neurokinin 1 receptor (NK1) antagonist for prevention of vomiting due to motion sickness in dogs.. |
PC-45396 |
NKP-608
|
A non-peptidic, specific, potent and orally active NK1 receptor antagonist with IC50 of 2.6 nM. |
PC-44659 |
SB-222200
|
A CNS-penetrant, potent and selective NK-3 receptor antagonist with Ki of 4.4 nM (inhibition of neurokinin B binding to CHO-hNK-3R). |