| Cat. No. |
Product Name |
Information |
| PC-42222 |
Y-39983
ROCK inhibitor
|
Y-39983 (Y-33075 hydrochloride) is a potent and selective p160 ROCK inhibitor with Ki of 140 nM. |
| PC-42541 |
Fasudil
ROCK inhibitor
|
Fasudil (AT-877, HA-1077) is a potent and selective inhibitor of Rho kinase (ROCK) with Ki of 0.33 uM (ROCK1). |
| PC-42540 |
Fasudil hydrochloride
ROCK inhibitor
|
Fasudil hydrochloride (AT-877, HA-1077) is a potent and selective inhibitor of Rho kinase (ROCK) with Ki of 0.33 uM (ROCK1). |
| PC-42776 |
GSK429286A
ROCK inhibitor
|
GSK429286A is a poten and selective inhibitor ROCK1 (IC50=14 nM) and ROCK2 (IC50=63 nM). |
| PC-22511 |
GNS-3595
ROCK2 inhibitor
|
GNS-3595 is a potent and selective ROCK2 inhibitor with IC50 of 5.7 nM, 80-fold selectivity over ROCK1 at 1mM ATP. |
| PC-22185 |
SB772077B dihydrochloride
ROCK inhibitor
|
SB772077B dihydrochloride (SB-772077B, SB77) is a potent, selective Rho kinase (ROCK) inhibitor with IC50 of 5.6 nM and 6.0 nM for ROCK1 and ROCK2, respectively. |
| PC-21755 |
C3TD879
Citron kinase inhibitor
|
C3TD879 is a potent, selective first-in-class Citron kinase (CITK) chemical inhibitor with biochemical IC50 of 12 nM. |
| PC-21300 |
ITRI-E-(S)4046
ROCK/MYLK4 inhibitor
|
ITRI-E-(S)4046 (E(S)4046) is a potent, highly specific, dual synergistic inhibitor of myosin light chain kinase 4 (MYLK4) and Rho-related protein kinase (ROCK) with IC50 of 3.2 nM and 25.6 nM for ROCK1 and MYLK4, respectively. |
| PC-20109 |
Y-33075 dihydrochloride
ROCK inhibitor
|
Y-33075 dihydrochloride (Y33075) is a potent, selective ROCK inhibitor with IC50 of 3.6 nM, more potent than Y-27632. |
