You are here:Home-Chemical Inhibitors & Agonists-GPCR-Sigma Receptor

Request The Product List ofSigma Receptor Sigma Receptor

Cat. No. Product Name Information
PC-49215

CT-189

Sigma 1 inhibitor

CT-189 (CT189) is a drug-like analog of IPAG and small-molecule Sigma1 receptor inhibitor, binds Sigma1 with Ki value of 38 nM in [3H](+)-pentazocine binding competition assays.
PC-47095

MAM03055A

Sigma 2 Receptor ligand

MAM03055A is a novel bivalent sigma-2 receptor/TMEM97 ligand with cytotoxic activity, exhibits high affinity and strong preference for sigma-2 receptor with Ki of 55.9 nM.
PC-38233

ANAVEX2-73

ANAVEX2-73 (Blarcamesine) is a Sigma-1 receptor agonist and muscarinic receptor modulator with neuroprotective effects.
PC-35305

BS148

Sigma 2 receptor agonist

BS148 (BS-148) is a potent, selective σ2 receptor agonist with pKi of 7.71, displays 25-fold selectivity over σ1.
PC-63494

JVW-1034

Sigma 2 Receptor ligand

JVW-1034 is a selective small molecule modulator of σ2R/Tmem97 with Ki of 23 nM, 10-fold weaker affinity for σ1R (Ki=248 nM).
PC-63432

Pridopidine

Pridopidine (ACR16, FR-310826, ASP-2314, Huntexil) is a selective and potent Sigma-1 receptor agonist.
PC-63205

MS-377

Sigma 1 receptor agonist

MS-377 is a potent, selective sigma-1 receptor ligand with Kd of 15.2 nM, showed anti-phencyclidine (PCP), anti-dopaminergic and anti-serotonergic activities.
PC-63203

E-5842

Sigma 1 receptor agonist

E-5842 (E5842) is a preferential sigma-1 receptor ligand, demonstrates potential atypical antipsychotic effects in vivo.
PC-63071

BD-1047 dihydrobromide

BD-1047 is a potent, selecitve Sigma 1 receptor (σ1) antagonist with Ki of 0.93 nM.
PC-63070

BD-1047

Sigma 1 receptor antagonist

BD-1047 is a potent, selecitve Sigma 1 receptor (σ1) antagonist with Ki of 0.93 nM.
PC-62223

Finazine

Sigma receptor ligand

Finazine is a high-affinity, brain penetrant sigma-1 and sigma 2 receptor ligand with Ki of 2.6 nM and 46 nM, respectively.
PC-61602

4-BBPB

Sigma 1 receptor agonist

4-BBPB is a highly potent agonist of sigma 1 receptor (σ1 receptor) with Ki of 0.8 nM.

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com