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Cat. No. Product Name Information
PC-45420

BD-1063 dhydrochloride

Sigma 1 receptor antagonist

BD-1063 dhydrochloride (BD1063) is a potent, selective sigma-1 receptor antagonist with binding Ki of 9 nM.
PC-45418

S1RA hydrochloride

Sigma 1 receptor antagonist

S1RA hydrochloride (E52862) is a potent and selective sigma-1 receptor (S1R) antagonist with Ki of 17 nM.
PC-45417

S1RA

Sigma 1 receptor antagonist

S1RA (E-52862) is a potent and selective sigma-1 receptor (S1R) antagonist with Ki of 17 nM.
PC-45419

PRE-084 hydrochloride

Sigma 1 receptor agonist

PRE-084 is a highly potent, selective sigma-1 receptor agonist with Ki of 2.2 nM, IC50 of 44 nM.
PC-42070

4-IBP

Sigma receptor agonist

4-IBP is a highly potent sigma receptor agonist with Ki of 1.7 nM and 25.2 nM for σ1 and σ2, respectively.
PC-24212

Cutamesine dihydrochloride

Sigma 1 receptor agonist

Cutamesine dihydrochloride (SA4503, AGY94806) is a potent, selective sigma 1 receptor (σ1R) agonist, shows igh affinity for sigma 1 receptor with IC50 of 17.4 nM, 100-fold over sigma 2 receptor.
PC-24211

SA4503

Sigma 1 receptor agonist

SA4503 (Cutamesine, AGY 94806) is a potent, selective sigma 1 receptor (σ1R) agonist, shows igh affinity for sigma 1 receptor with IC50 of 17.4 nM, 100-fold over sigma 2 receptor.
PC-24026

Fabomotizole hydrochloride

Sigma 1 receptor agonist

Fabomotizole hydrochloride (Afobazole, CM346) is a compound with anxiolytic and neuroprotective activities, is an agonist of sigma1-receptor (S1R, Ki=5.9 uM).
PC-24025

Afobazole

Sigma 1 receptor agonist

Afobazole (Fabomotizole, CM346) is a compound with anxiolytic and neuroprotective activities, is an agonist of sigma1-receptor (S1R, Ki=5.9 uM).
PC-23425

Amylovis-201

Sigma-1 agonist

Amylovis-201 is dual-target ligand acting as an anti-amyloidogenic compound and a potent agonist of the σ1 chaperone protein, interferes with Amyloid-β aggregation.
PC-22349

WLB-87848

Sigma 1 receptor agonist

WLB-87848 is a highly potent, selective, orally bioavailable sigma-1 receptor (σ1R) agonist with Ki of 9 nM, with ni significant affinity for σ2R.
PC-21111

AZ-66

Sigma receptor antagonist

AZ-66 is a highly potent S1R/S2R antagonist with Ki of 0.31/1.76 nM, respectively.

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