| Cat. No. |
Product Name |
Information |
| PC-22031 |
TIM-098a
AAK1 inhibitor
|
TIM-098a is a potent, selective AP2-associated protein kinase 1 (AAK1) with IC50 of 0.24 uM, inhibits AAK1 activity in transfected cultured cells with IC50 of 0.87 uM. |
| PC-20649 |
BMS-911172
AAK1 inhibitor
|
BMS-911172 is a potent, selective and brain penetrant adaptor protein 2-associated kinase 1 (AAK1) inhibitor with IC50 of 12 nM. |
| PC-72847 |
LX9211
AAK1 inhibitor
|
LX9211 (BMS-9861761) is a highly selective, CNS-penetrable, and potent AAK1 inhibitor with IC50 of 2.0 nM. |
| PC-35961 |
AAK1 inhibitor 25A
AAK1 inhibitor
|
AAK1 inhibitor 25A is a potent, selective inhibitor of AAK1 and the closely related kinase BMP2K with Ki of 8 nM (AAK1). |
| PC-35853 |
SGC-AAK1-1
AAK1 inhibitor
|
AAK1 inhibitor 1 (SGC-AAK1-1) is a potent, selective inhibitor of AAK1 and BMP2K/BIKE ((BMP-2 inducible kinase)) that potently targets the ATP-binding site (AAK1 Ki =9.1 nM, BIKE Ki= 17 nM). |
| PC-35098 |
BMT-046091
AAK1 inhibitor
|
BMT-046091 (BMT046091) is a potent and selective AAK1 inhibitor with IC50 of 2.8 nM. |
| PC-60637 |
BMS-901715
AAK1 inhibitor
|
BMS-901715 (BMS901715) is a potent, selective adapter protein-2 associated kinase 1 (AAK1) inhibitor with IC50 of 3.3 nM. |
| PC-60636 |
BMT-090605
AAK1 inhibitor
|
BMT-090605 (BMT 090605, BMT090605) is a potent, selective adapter protein-2 associated kinase 1 (AAK1) inhibitor with IC50 0.6 nM. |
| PC-60635 |
LP-935509
AAK1 inhibitor
|
LP-935509 (LP935509) is a potent, selective and brain-penetrant adapter protein-2 associated kinase 1 (AAK1) inhibitor with IC50 of 3.3 nM. |
| PC-23576 |
HW161023
AAK1 inhibitor
|
HW161023 is a potent, selective AAK1 inhibitor with IC50 of 5.4 nM. |
| PC-20650 |
AAK1 inhibitor (S)-31
AAK1 inhibitor
|
AAK1 inhibitor (S)-31 is a potent, selective and brain penetrant adaptor protein 2-associated kinase 1 (AAK1) inhibitor with IC50 of 5.8 nM. |
