| Cat. No. |
Product Name |
Information |
| PC-21883 |
(+)-JJ-74-138
Androgen Receptor inhibitor
|
(+)-JJ-74-138 is a non-competitive androgen receptor (AR) antagonist, directly interacts with AR with SPR KD of 4.29 uM, inhibits AR with mutations in the LBD or lacking ligand binding domain (LBD). |
| PC-21502 |
AR inhibitor 1ae
AR inhibitor
|
AR inhibitor 1ae is a small-molecule inhibitor of the androgen receptor activation domain (AR AD) with IC50 of 1.54 uM in androgen-induced PSA-luciferase assays, inhibits AR-V7 transcriptional activity with IC50 of 4.1 uM. |
| PC-21405 |
UT-34
AR inhibitor
|
UT-34 is a potent, second-generation androgen receptor (AR) pan antagonist, degrades enzalutamide-sensitive and -resistant ARs and AR splice variants (AR-SVs). |
| PC-21404 |
UT-105
AR inhibitor
|
UT-105 is a small-molecule, irreversible, selective androgen receptor (AR) degrader (SARD) and irreversible inhibitor, binds to AR N-terminal domain (NTD) and inhibits both the AR and AR splice variants (AR-SVs). |
| PC-20797 |
M17-B15
AR inhibitor
|
M17-B15 is a potent, specific small molecule inhibitor of androgen receptor (AR) targeting the dimer interface pocket (DIP), inhibits AR transcriptional inhibition with IC50 of 0.03 uM. |
| PC-35497 |
Leelamine hydrochloride
|
Leelamine hydrochloride (Dehydroabietylamine) is a novel inhibitor of androgen receptor (AR), inhibits castration-resistant prostate cancer cells. |
| PC-45255 |
Boldenone undecylenate
|
A synthetic, anabolic-androgenic steroid (AAS) and androgen ester that is used in veterinary medicine, a long-acting ester of boldenone.. |
