| Cat. No. |
Product Name |
Information |
| PC-43002 |
Trenbolone acetate
|
Trenbolone acetate (RU-1697,17beta-TBOH) is a potent testosterone analog and selective androgen receptor modulator, is an androgen ester and a long-acting prodrug of trenbolone. |
| PC-42895 |
BMS-564929
SARM
|
BMS-564929 is a potent, selective androgen receptor modulator (SARM) that binds to AR with Ki of 2.11 nM. |
| PC-42838 |
Andarine
SARM
|
Andarine (S4, GTx007) is a non-steroidal selective androgen receptor modulator (SARM) with Ki of 4 nM, efficaciously stimulates AR-mediated reporter gene expression. |
| PC-62000 |
Enobosarm
SARM
|
Enobosarm (GTx-024, MK-2866, Ostarine) is a selective androgen receptor modulator (SARM) for the treatment of conditions such as muscle wasting and osteoporosis. |
| PC-61999 |
LY2452473
SARM
|
LY2452473 (TT 701, OPK 88004) is an orally bioavailable selective androgen receptor modulator (SARM) being developed for the treatment of disorders related to hypogonadism. |
| PC-61861 |
LGD-3303
SARM
|
LGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors. |
| PC-61774 |
VPC14449
AR DBD inhibitor
|
VPC14449 (VPC-14449) is a potent and selective androgen receptor DNA-binding domain (AR-DBD) inhibitor with IC50 of 0.34 uM, without affecting AR protein expression. |
| PC-61678 |
EPI-001
AR NTD inhibitor
|
EPI-001 is a small molecule that blocks transactivation of the androgen Receptor (AR) NTD (IC50=6 uM) and specificly inhibits AR without attenuating transcriptional activities of related steroid receptors. |
| PC-61444 |
Metribolone
AR ligand
|
Metribolone (R1881) is an orally active anabolic-androgenic steroid and a 19-nortestosterone derivative that has been widely used in scientific research as a hot ligand in androgen receptor (AR) ligand binding assays (LBAs) and as a photoaffinity label for the AR. |
| PC-61086 |
BMS-641988
AR antagonist
|
BMS-641988 is a potent, selective, nonsteroidal androgen receptor antagonist with Ki of 1.7 nM, MDA-MB-453 cell IC50 of 16 nM. |
| PC-60530 |
Ralaniten acetate
AR-NTD inhibitor
|
Ralaniten acetate (EPI-506) is the acetate prodrug of Ralaniten (EPI-002), a small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer. |
| PC-60529 |
Ralaniten
AR-NTD inhibitor
|
Ralaniten (EPI-002) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor, inhibits AR transcriptional activity with IC50 of 7.4 uM. |
