| Cat. No. |
Product Name |
Information |
| PC-61444 |
Metribolone
AR ligand
|
Metribolone (R1881) is an orally active anabolic-androgenic steroid and a 19-nortestosterone derivative that has been widely used in scientific research as a hot ligand in androgen receptor (AR) ligand binding assays (LBAs) and as a photoaffinity label for the AR. |
| PC-61086 |
BMS-641988
AR antagonist
|
BMS-641988 is a potent, selective, nonsteroidal androgen receptor antagonist with Ki of 1.7 nM, MDA-MB-453 cell IC50 of 16 nM. |
| PC-60530 |
Ralaniten acetate
AR-NTD inhibitor
|
Ralaniten acetate (EPI-506) is the acetate prodrug of Ralaniten (EPI-002), a small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer. |
| PC-60529 |
Ralaniten
AR-NTD inhibitor
|
Ralaniten (EPI-002) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer. |
| PC-70129 |
Proxalutamide
AR antagonist
|
Proxalutamide (GT-0918) is a potent androgen receptor (AR) antagonist with ability to down regulate AR protein level in prostate cancer cells. |
| PC-70118 |
LGD4033
SARM
|
LGD-4033 (VK-5211, Ligandrol) is a nonsteroidal, oral selective androgen receptor modulator (SARM), binds androgen receptor with high affinity (Ki=1 nM) and selectivity. |
| PC-45422 |
GLPG-0492 R enantiomer
|
The R enantiomer of GLPG-0492, a non-steroidal selective androgen receptor modulator (SARM) for treatment for Duchenne muscular dystrophy (DMD). |
| PC-45612 |
ORM-15341
AR inhibitor
|
ORM-15341 (Ketodarolutamide, BAY1896953) is the active main metabolite of ODM-201, a potent wt/mutant androgen receptor (AR) inhibitor, inhibits wtAR/AR(F876L) with IC50s of 25/51 nM respectively. |
| PC-45932 |
Enzalutamide
AR antagonist
|
Enzalutamide (MDV3100) is a potent, selective and orally available androgen-receptor (AR) antagonist with IC50 of 36 nM. |
| PC-42794 |
MK-0773
SARM
|
MK-0773 (PF-05314882) is a potent, selective androgen receptor modulator (SARM) with binding IC50 of 6.6 nM. |
| PC-45113 |
ODM-201
AR antagonist
|
ODM-201 (BAY-1841788, Darolutamide) is a potent wt/mutant androgen receptor (AR) inhibitor with Ki of 11 nM. |
| PC-42075 |
GSK2881078
SARM
|
GSK2881078 potent and selective androgen receptor modulator (SARM), act as partial AR agonist and induces AR-mediated transcriptional activation in PC3(AR)2 cells with EC50 of 3.99 nM. |
