Cat. No. |
Product Name |
Information |
PC-21943 |
MRK-898
GABA A modulator
|
MRK-898 is an orally active GABA(A) receptor modulator, binds to α1, α2, α3 or α5 subunit of GABA(A) receptor with Ki values of 1.2 nM, 1.0 nM, 0.73 nM, and 0.50 nM, respectively. |
PC-21611 |
DS-II-73
GABAAR modualtor
|
DS-II-73 is a selective α2/3/5-containing GABAA receptor (GABAAR) potentiator with IC50 of 320 nM, 381 nM and 435 nM for α2β3γ2 α3β3γ2 α5β3γ2. |
PC-42115 |
DMCM hydrochloride
|
A potent benzodiazepine inverse agonist that displays anxiogenic and potent convulsant activity. |
PC-45152 |
Acamprosate calcium
|
A GABA receptor agonist and modulator of glutamatergic systems. |
PC-45172 |
(R)-Baclofen hydrochloride
|
A derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist. |
PC-42068 |
Pipequaline
|
A clinically-effective anxiolytic that acts as a non-selective partial agonist of benzodiazepine receptor. |