| Cat. No. |
Product Name |
Information |
| PC-42106 |
PK-14105
|
A potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM. |
| PC-45592 |
Indiplon
|
A potent GABAA receptor positive allosteric modulator that acts at the benzodiazepine site (Ki values are 1.2 and 1.7 nM in rat frontal cortex and cerebellum respectively). |
| PC-42225 |
U-93631
|
A potent GABAA receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction. |
| PC-42115 |
DMCM hydrochloride
|
A potent benzodiazepine inverse agonist that displays anxiogenic and potent convulsant activity. |
| PC-45628 |
Lorediplon
|
A partial positive allosteric GABAA receptor modulator. |
| PC-45060 |
Basmisanil
|
A novel selective negative allosteric modulator of the GABAA receptor α5-subtype, which is under development for the treatment of cognitive impairment associated with Down syndrome.. |
| PC-45152 |
Acamprosate calcium
|
A GABA receptor agonist and modulator of glutamatergic systems. |
| PC-46124 |
Baclofen
|
A derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist. |
| PC-45172 |
(R)-Baclofen hydrochloride
|
A derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist. |
| PC-45171 |
(R)-Baclofen
|
A derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist. |
| PC-42068 |
Pipequaline
|
A clinically-effective anxiolytic that acts as a non-selective partial agonist of benzodiazepine receptor. |
