| Cat. No. |
Product Name |
Information |
| PC-20260 |
AZD-5423
GR modulator
|
AZD-5423 (AZD5423) is a potent, nonsteroidal, selective glucocorticoid receptor modulator with IC50 of 49 pM for inhibition of AP-1 mediated transcription. |
| PC-73325 |
LEO 134310
GR agonist
|
LEO 134310 (LP 0155) is a non-steroidal, potent and selective glucocorticoid receptor (GR) agonist (EC50=2 nM, hPBMC). |
| PC-72993 |
OP-3633
GR antagonist
|
OP-3633 (OP3633) is a potent and selective steroidal glucocorticoid receptor (GR) antagonist with an IC50 of 29 nM. |
| PC-38103 |
Glucocorticoid receptor modulator-1
GR modulator
|
Glucocorticoid receptor modulator-1 is a glucocorticoid receptor modulator.. |
| PC-35571 |
ORIC-101
Glucocorticoid receptor inhibitor
|
ORIC-101 (ORIC101) is a highly potent, selective steroidal glucocorticoid receptor (GR) antagonist (IC50=5.6 nM) with reduced androgen receptor (AR) agonistic activity. |
| PC-35449 |
Exicorilant
|
Exicorilant (CORT125281, CORT-125281) is a potent, selective glucocorticoid receptor (GR) antagonist, exhibits no cross-reactivity for the PR and AR receptors.. |
| PC-63143 |
AZD-7594
|
AZD-7594 (AZ-13189620) is a potent, nonsteroidal, selective glucocorticoid receptor modulator (SGRM) with binding IC50 of 0.9 nM, shows no affinity for AR, PR, MR and ERα/β. |
| PC-61603 |
Mapracorat
|
Mapracorat (ZK 245186) is a potent, selective and non-steroid glucocorticoid receptor (GR) agonist with binding Ki of 1.9 nM. |
| PC-60801 |
LLY-2707
|
LLY-2707 (LLY 2707, LLY2707) is a novel potent, selective, nonsteroidal glucocorticoid receptor antagonist with Ki of 2.13 nM. |
| PC-60072 |
AZD-9567 monohydrate
|
AZD-9567 monohydrate is a potent, selective, non-steroidal and orally available selective glucocorticoid receptor modulator (SGRM) for treatment of rheumatoid arthritis.. |
| PC-60071 |
AZD-9567
|
AZD-9567 (AZD9567) is a potent, selective, non-steroidal and orally available selective glucocorticoid receptor modulator (SGRM) for treatment of rheumatoid arthritis.. |
| PC-45178 |
Loteprednol etabonate
|
Loteprednol etabonate is an anti-inflammatory corticosteroid used in optometry and ophthalmology. |
