Cat. No. |
Product Name |
Information |
PC-23473 |
JNJ-7777120
H4R antagonist
|
JNJ-7777120 (JNJ 7777120) is potent and selective histamine H4 receptor (H4R) antagonist with Ki of 4.5 nM (hH4R), >1000-fold selectivity over H1, H2, or H3 receptors. |
PC-23262 |
Izuforant
H4R antagonist
|
Izuforant (JW1601, LEO 152020) is a potent, selective and oral histamine 4 receptor (H4R) antagonist with IC50 of 65.1-72.2 nM in human whole-blood assay, and pKi of 6.83 and 5.36 at mouse and rat histamine receptor subtypes. shows lower pKi values against other histamine receptor. |
PC-42910 |
Pitolisant oxalate
|
A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM. |