| Cat. No. |
Product Name |
Information |
| PC-35982 |
SUVN-G3031 free base
H3R inverse agonist
|
SUVN-G3031 (Samelisant) free base is a potent, selective, orally active histamine H3 receptor (H3R) inverse agonist with Ki of 8.73 nM (hH3R). |
| PC-35981 |
SUVN-G3031
H3R inverse agonist
|
SUVN-G3031 (Samelisant) is a potent, selective, orally active histamine H3 receptor (H3R) inverse agonist with Ki of 8.73 nM (hH3R). |
| PC-35408 |
JNJ-5207852
Histamine H3 antagonist
|
JNJ-5207852 (JNJ5207852) is a potent, selective antagonist of H3 receptor with pKi of 8.9 and 9.24 for rat and human H3, respectively. |
| PC-35407 |
Contilisant
AChE inhibitor
|
Contilisant is a neuroprotective, non-toxic, antioxidant, permeable ligand, showing in vitro pharmacological properties on the selected biological targets (hAChE IC50=0.53 uM. |
| PC-35223 |
Clobenpropit dihydrobromide
Histamine H3 inverse agonist
|
Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors. |
| PC-35222 |
Clobenpropit
Histamine H3 antagonist
|
Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors. |
| PC-63422 |
UR-PI376
Histamine H4 agonist
|
UR-PI376 is a potent, selective histamine H4 receptor (hH4R) agonist with pEC50 of 7.47, shows negligible hH1R and hH2R activities and significant selectivity over the hH3R.. |
| PC-63421 |
OUP-16
Histamine H4 agonist
|
OUP-16 is a potent H4R agonist with a considerable selectivity over H3R. |
| PC-63420 |
A-943931
Histamine H4 antagonist
|
A-943931 is a potent, selective antagonist of histamine H4 receptor (H4R) with binding pKi of 8.33 and 8.42 for hH4 and rH4, respectively. |
| PC-63419 |
A-943931 dihydrochloride
Histamine H4 antagonist
|
A-943931 dihydrochloride is a potent, selective antagonist of histamine H4 receptor (H4R) with binding pKi of 8.33 and 8.42 for hH4 and rH4, respectively. |
| PC-63418 |
VUF 10214
Histamine H4 ligand
|
VUF-10214 is a potent, selective histamine H4 receptor (H4R) ligand with pKi of 7.4, shows anti-inflammatory properties in vitro. |
| PC-63417 |
JNJ-40279486
Histamine H4 antagonist
|
JNJ-40279486 is a potent, selective histamine H4 receptor antagonist with Ki of 9.4 nM (hH4), demonstrates acceptable pharmacokinetic profile and efficacy in mouse model of inflammation.. |
