| Cat. No. |
Product Name |
Information |
| PC-61337 |
MK-7288
|
A novel histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome. |
| PC-60793 |
JNJ 39758979
|
A potent, selective, orally bioavailable histamine H4 receptor antagonist with Ki of 12.5 nM, >80-fold selectivity over other histamine receptors. |
| PC-60738 |
AZD 3676
|
A novel potent, combined serotonin 5-HT1A and 5-HT1B receptor antagonist with Ki of 0.13 and 2.4 nM in brain homogenates, respectively. |
| PC-60377 |
S-38093
|
A novel brain-penetrant H3 receptor antagonist/inverse agonist that shows procognitive properties in vivo. |
| PC-45168 |
Loratadine
|
A tricyclic antihistamine that acts as a selective inverse agonist of peripheral histamine H1-receptors.. |
| PC-45167 |
Cetirizine dihydrochloride
|
A second-generation antihistamine that acts as a selective H1 receptor antagonist. |
| PC-45166 |
Cetirizine
|
A second-generation antihistamine that acts as a selective H1 receptor antagonist. |
| PC-42380 |
VUF10460
|
A potent, selective histamine H4 receptor agonist with pKi of 7.46 and 8.22 for rat and human H4, respectively. |
| PC-42908 |
ABT-239
|
A potent and selective Histamine H3 receptor antagonist with Ki of 0.1-5.8 nM (human, rat H3). |
| PC-42911 |
Pitolisant hydrochloride
|
A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM. |
| PC-42910 |
Pitolisant oxalate
|
A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM. |
| PC-45163 |
Alcaftadine
|
A H1 histamine receptor antagonist that used for prevention of allergic conjunctivitis.. |
