| Cat. No. |
Product Name |
Information |
| PC-72277 |
Enerisant hydrochloride
H3R antagonist
|
Enerisant hydrochloride (TS091 hydrochloride) is a potent, selective histamine H3 receptor antagonist/inverse agonist with IC50 of 2.89 and 14.5 nM against hH3R and rH3R, respectively. |
| PC-72276 |
Enerisant
H3R antagonist
|
Enerisant (S091,TS-091) is a potent, selective histamine H3 receptor antagonist/inverse agonist with IC50 of 2.89 and 14.5 nM against hH3R and rH3R, respectively. |
| PC-36027 |
K-8986 maleate
|
K-8986 maleate (K8986) is a histamine H1-receptor antagonist with potential therapeutic for treatment of allergic conjunctivitis.. |
| PC-35408 |
JNJ-5207852
|
JNJ-5207852 (JNJ5207852) is a potent, selective antagonist of H3 receptor with pKi of 8.9 and 9.24 for rat and human H3, respectively. |
| PC-35407 |
Contilisant
|
Contilisant is a neuroprotective, non-toxic, antioxidant, permeable ligand, showing in vitro pharmacological properties on the selected biological targets (hAChE IC50=0.53 uM. |
| PC-35222 |
Clobenpropit
|
Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors. |
| PC-63421 |
OUP-16
|
OUP-16 is a potent H4R agonist with a considerable selectivity over H3R.. |
| PC-63419 |
A-943931 dihydrochloride
|
A-943931 dihydrochloride is a potent, selective antagonist of histamine H4 receptor (H4R) with binding pKi of 8.33 and 8.42 for hH4 and rH4, respectively. |
| PC-63418 |
VUF-10214
|
VUF-10214 is a potent, selective histamine H4 receptor (H4R) ligand with pKi of 7.4, shows anti-inflammatory properties in vitro.. |
| PC-63413 |
JNJ-28610244
|
JNJ-28610244 is a potent, selective agonist of histamine H4 receptor (H4R).. |
| PC-63410 |
JNJ-28307474
|
JNJ-28307474 is a potent, selective antagonist of the histamine H4 receptor (H4R), inhibits LPS-induced TNF production.. |
| PC-63401 |
JNJ-18038683 free base
|
JNJ-18038683 is a potent, selective 5-HT7 receptor antagonist with pKi of 8.19 and 8.20 for rat and human 5-HT7 in cell-based assays. |
