| Cat. No. |
Product Name |
Information |
| PC-61615 |
Irdabisant
H3 receptor antagonist
|
Irdabisant (CEP-26401) is a potent, selective, orally active histamine H3 receptor antagonist with Ki of 2 nM and 7 nM for human and rat H3Rs, respectivity. |
| PC-61569 |
Burimamide oxalate
H3/H2 receptor antagonist
|
Burimamide oxalate is a potent dual H3/H2 receptor antagonist with Ki of 0.07 and 7.8 uM, respectively. |
| PC-61568 |
Burimamide
H3/H2 receptor antagonist
|
Burimamide is a potent dual H3/H2 receptor antagonist with Ki of 0.07 and 7.8 uM, respectively. |
| PC-61567 |
Adriforant
Histamine H4 antagonist
|
Adriforant (PF-3893787, ZPL 3893787) is a potent and selective H4 receptor antagonist with binding Ki of 2.4 nM. |
| PC-61562 |
APD916
Histamine H3 antagonist
|
APD916 is a potent and selective antagonist of the H3 receptor with Ki of 0.7 nM for rH3R. |
| PC-61337 |
MK-7288
H3R inverse agonist
|
MK-7288 is a selective histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome. |
| PC-60793 |
JNJ-39758979
Histamine H4 antagonist
|
JNJ-39758979 is a potent, selective, orally bioavailable histamine H4 receptor antagonist with Ki of 12.5 nM, >80-fold selectivity over other histamine receptors. |
| PC-60533 |
Seliforant
Histamine H4 antagonist
|
Seliforant (SENS-111, SENS111) is a novel potent, selective histamine H4 receptor antagonist. |
| PC-60377 |
S 38093
Histamine H3 antagonist
|
S 38093 is a brain-penetrant H3 receptor antagonist/inverse agonist that shows procognitive properties in vivo. |
| PC-45168 |
Loratadine
Histamine H1 agonist
|
A tricyclic antihistamine that acts as a selective inverse agonist of peripheral histamine H1-receptors.. |
| PC-45167 |
Cetirizine dihydrochloride
Histamine H1 antagonist
|
Cetirizine dihydrochloride is a second-generation antihistamine that acts as a selective H1 receptor antagonist, inhibits eosinophil chemotaxis during the allergic response. |
| PC-45166 |
Cetirizine
Histamine H1 antagonist
|
Cetirizine is a second-generation antihistamine that acts as a selective H1 receptor antagonist, inhibits eosinophil chemotaxis during the allergic response. |
