| Cat. No. |
Product Name |
Information |
| PC-63399 |
Toreforant
|
Toreforant (JNJ-38518168) is a potent, selective histamine H4 receptor (H4R) antagonist with Ki of 8.4 nM, shows excellent selectivity over other receptors including the other histamine receptors. |
| PC-63034 |
PF-03654746
|
PF-03654746 (PF 3654746) is a potent, selective, orally bioactive antagonist of H3 receptor with Ki of 2.3 nM. |
| PC-63033 |
PF-03654764
|
PF-03654764 (PF 3654764) is a potent, selective, orally bioactive antagonist of H3 receptor with Ki of 1.4 nM. |
| PC-63032 |
ABT-288
|
ABT-288 is a potent, selective and competitive antagonist of H3 receptor with Ki of 1.9/8.2 nM for human/rat H3 respectively. |
| PC-61996 |
LY2624803
|
LY2624803 is a novel potent histamine H1 and 5HT-2A receptor modulator in the pipeline for treating insomnia.. |
| PC-61663 |
JNJ 10181457 dihydrochloride
|
JNJ 10181457 is a neutral, potent and selective, brain penetrant H3 antagonist with pKi of 8.93, pA2 of 9.22 for hH3. |
| PC-61662 |
JNJ 10181457
|
JNJ 10181457 is a neutral, potent and selective, brain penetrant H3 antagonist with pKi of 8.93, pA2 of 9.22 for hH3. |
| PC-61661 |
JNJ 39220675
|
JNJ 39220675 is potent and selective, brain penetrant H3 antagonist with Ki of 1.4 nM, pA2 of 9.42 for hH3. |
| PC-61616 |
Irdabisant hydrochloride
|
Irdabisant (CEP-26401) is a potent, selective, orally active histamine H3 receptor antagonist with Ki of 2 nM and 7 nM for human and rat H3Rs, respectivity. |
| PC-61569 |
Burimamide oxalate
|
Burimamide oxalate is a potent dual H3/H2 receptor antagonist with Ki of 0.07 and 7.8 uM, respectively. |
| PC-61568 |
Burimamide
|
A potent dual H3/H2 receptor antagonist with Ki of 0.07 and 7.8 uM, respectively. |
| PC-61562 |
APD916
|
APD916 is a potent and selective antagonist of the H3 receptor with Ki of 0.7 nM for rH3R. |
