Cat. No. |
Product Name |
Information |
PC-23064 |
GNE-6893
HPK1 inhibitor
|
GNE-6893 is a potent, selective and orally active inhibitor of HPK1 (hematopoietic progenitor kinase 1) with Ki of <0.019 nM, potently inhibits phosphorylation of SLP76 with IC50 of 44 nM in Jurkat cell assay. |
PC-22569 |
HPK1-IN-3
HPK1 inhibitor
|
HPK1-IN-3 is a potent, selective, ATP-competitive hematopoietic progenitor kinase 1 (HPK1, MAP4K1) inhibitor with IC50 of 0.25 nM in TR-FRET assays. |
PC-22568 |
KHK-6
HPK1 inhibitor
|
KHK-6 is a potent, selective, ATP-competitive inhibitor of serine/threonine kinase hematopoietic progenitor kinase 1 (HPK1, MAP4K1) with IC50 of 20 nM. |