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Cat. No. Product Name Information
PC-38142

SBI-553

NTR1 modulator

SBI-553 (SBI553) is a potent, selective, β-arrestin-biased, brain penetrant neurotensin receptor 1 (NTR1, NTSR1) allosteric modulator with EC50 of 0.34 uM.
PC-61109

NTRC-844

NTRC-844 (NTRC844) is a potent, selective neurotensin receptor type 2 (NTS2) with Ki of 23 nM, 100-fold selectivity over NTS1 receptor.
PC-60948

SR142948

SR142948 is a potent, selective and orally active neurotensin receptor antagonist with IC50 of 1.19 nM.
PC-20497

SR142948 hydrochloride

NT receptor antagonist

SR142948 hydrochloride is a potent, selective and orally active neurotensin receptor antagonist with IC50 of 1.19 nM.
PC-20496

JMV449

NTR1 agonist

JMV449 (JMV-449) is a potent, metabolically stable neurotensin receptor agonist peptide with IC50 of 0.15 nM for inhibition of [125I]-NT binding to neonatal mouse brain.
PC-20493

ML314

NTR1 agonist

ML314 is a selective, brain penetrant full agonist of neurotensin 1 receptor (NTR1) with EC50 of 2.0 uM, shows good selectivity against NTR2 and GPR35.
PC-20492

ML301

NTR1 agonist

ML301 is a selective full (79-93%) neurotensin-1 (NTR1) receptor agonist with EC50 of 2.0-4.1 uM, good selectivity relative to NTR2 and GPR35.
PC-60947

SR 48692

A potent, selective and orally active nonpeptide antagonist of the neurotensin receptor with IC50 of 0.99 nM (guinea pig), without any intrinsic agonist activity.

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