| Cat. No. |
Product Name |
Information |
| PC-61432 |
STX681
Aromatase/Steroid sulfatase inhibitor
|
STX681 is a potent, orally active, dual-acting aromatase and steroid sulfatase (STS) inhibitor with IC50 of 0.82 nM and 39 nM, respectively. |
| PC-61431 |
Irosustat
|
Irosustat (STX-64, BN-83495, Oristusane, 667-coumate) is an orally active, highly potent, irreversible, nonsteroidal inhibitor of steroid sulfatase (STS) with IC50 of 8 nM. |
| PC-61435 |
Estrone sulfamate
|
A potent, irreversible, and orally active inhibitor of steroid sulfatase (STS) with IC50 of 65 pM in intact MCF-7 cells. |
| PC-61434 |
KW-2581
|
A novel potent, irreversible and orally active inhibitor of steroid sulfatase (STS) with IC50 of 13 nM in ZR-75-1 cells. |
| PC-61433 |
SR-16157
|
A novel dual-acting steroid sulfatase inhibitor (IC50=0.1 uM) and selective ERα modulator (SERM). |
| PC-61430 |
STX-213
|
An orally active, second-generation steroid sulfatase inhibitor with IC50 of 0.5 nM. |
