| Cat. No. |
Product Name |
Information |
| PC-72628 |
Ralmitaront
TAAR1 modulator
|
Ralmitaront (RO6889450, RG7906) is a potent, orally active trace amine-associated receptor 1 (TAAR-1) modulator as a neuroleptic agent. |
| PC-72627 |
Ulotaront
TAAR1 agonist
|
Ulotaront (SEP-363856, SEP-856) is a novel psychotropic agent with agonism at trace amine receptor 1 (TAAR1) and 5-HT1A receptors but no appreciable action at dopamine D2 receptors. |
| PC-61078 |
Alpha-NETA free base
|
Alpha-NETA is a selective choline acetyltransferase (ChA) inhibitor with IC50 of 9 uM, also is a TAAR5 agonist that affects sensory gating in rats. |
| PC-61077 |
RO 5203648
|
RO 5203648 is a potent and selective TAAR1 partial agonist with Ki of 0.5, 1.0, 6.8 and 2.6 nM for mouse, rat, human and monkey TAAR1, respectively. |
| PC-61075 |
RO 5166017
TAAR1 agonist
|
RO 5166017 is a potent, selective TAAR1 agonist with Ki of 1.9, 2.7, 31 and 24 nM for mouse, rat, cynomolgus monkey and human TAAR1 stably expressed in HEK293 cells. |
| PC-61073 |
EPPTB
|
EPPTB (RO5212773) is a potent, selective mouse TAAR1 antagonist that potently antagonizes cAMP production induced by 1.5 uM β-phenylethylamine with IC50 of 27.5 nM, Ki of 1 nM. |
| PC-61072 |
RO 5263397
TAAR1 agonist
|
RO 5263397 is a highly potent, selective and orally bioavailable trace amine-associated receptor 1 (TAAR1) partial agonist with EC50 of 17 nM, >1,000-fold selectivity over human adrenergic α2A receptor. |
| PC-72353 |
RTI-7470-44
hTAAR1 antagonist
|
RTI-7470-44 is a potent, selective human trace amine-associated receptor subtype 1 (hTAAR1) inhibitor with IC50 of 8.4 nM in vitro cAMP functional assay. |
| PC-61076 |
RO 5073012
|
A potent, selective, orally active TAAR1 partial agonist with Ki of 6 nM, EC50 of 23 nM (hTAAR1), 140-fold selectivity over β2 adrenergic receptors. |
| PC-61074 |
Ractopamine
|
A small molecule TAAR1 agonist and β adrenoreceptor agonist that stimulates β1 and β2 adrenergic receptors. |
| PC-61071 |
RO 5256390
|
A highly potent, selective and orally bioavailable trace amine-associated receptor 1 (TRRA1) full agonist with EC50 of 18 nM, >500-fold selectivity over human adrenergic α2A receptor. |
