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Cat. No. Product Name Information
PC-49652

OPC-61815

V2R inhibitor

OPC-61815 (Tolvaptan phosphate ester sodium) is a water-soluble phosphate ester pro-drug of Tolvaptan (Cat# PC-45125), which is an orally active vasopressin V2 receptor antagonist.
PC-38647

Enuvaptan

V1AR antagonist

Enuvaptan (BAY2327949) is a potent, selective vasopressin 1a receptor (V1AR) antagonist with potential for renal and cardiovascular diseases.
PC-36095

Pecavaptan

V1a/V2 receptor antagonist

Pecavaptan (BAY 1753011) is a potent, orally active and dual antagonist of vasopressin receptor V1a/V2 receptor (Ki=0.5 nM and 0.6 nM for human, respectively).
PC-62116

ML389

V1AR antagonist

ML389 is a highly potent, selective vasopressin receptor 1a (V1a-R) antagonist with IC50 of 40 nM.
PC-61507

TASP0434299

V1BR radioligand

TASP0434299 is a radioligand candidate for arginine vasopressin 1B (V1B) receptor that exhibits high binding affinities for human and rat V1B receptors with IC50 of 0.526 and 0.641 nM, respectively.
PC-70166

Conivaptan

Vasopressin Receptor inhibitor

Conivaptan (YM-087) is a potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively.
PC-60078

RG7713

V1a receptor antagonist

RG7713 (RO5028442, RG-7713) is a potent, highly selective, brain-penetrant vasopressin 1a (hV1a) antagonist with Ki of 1 nM.
PC-60033

Balovaptan

V1a receptor antagonist

Balovaptan (RG7314, RO5285119) is a potent, selective vasopressin-1 receptor antagonist with Kb of 0.39 nM at the human V1a receptor.
PC-47487

Ornipressin

Ornipressin is a vasoconstrictor, haemostatic and renal agent.
PC-45192

Desmopressin

V2 receptor antagonist

Desmopressin is a synthetic analogue of the antidiuretic hormone arginine vasopressin, binds to V2 receptors in renal collecting ducts, increasing water reabsorption.
PC-45191

Desmopressin acetate

Desmopressin acetate is a synthetic analogue of the antidiuretic hormone arginine vasopressin.
PC-45459

Mozavaptan

V2 receptor antagonist

Mozavaptan (OPC-31260) is a potent, selective nonpeptide vasopressin V2 receptor antagonist with IC50 of 14 nM.

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