| Cat. No. |
Product Name |
Information |
| PC-21153 |
GPR55 agonist 28
GPR55 agonist
|
GPR55 agonist 28 is a potent, selective GPR55 agonist with EC50 of 131 and 141 nM for human and rat GPR55, respectively, in Ca2+ flux assays. |
| PC-20401 |
ML192
GPR55 inhibitor
|
ML192 (CID1434953) is a potent, selective antagonist of GPR55 with IC50 of 1080 nM, >45-fold antagonist and agonist selectivity against GPR35, CB1 and CB2. |
| PC-38506 |
PSB-SB-487
GPR55 inhibitor
|
PSB-SB-487 is a potent, selective antagonist of orphan G-protein-coupled receptor GPR55 with IC50 value 113 nM, and KB value 561 nM (hGPR55), shows little to no activity against CB1/CB2 and GPR18 receptors. |
| PC-38003 |
(R,S)-MNF
GPR55 inhibitor
|
(R,S′)-MNF is a bi-functional GPR55 inhibitor and biased β2 adrenergic agonist, inhibits proliferation of PDAC cell lines (IC50=0.11 uM, PANC-1 cells). |
| PC-35196 |
O-1602
GPR55 agonist
|
O-1602 (O1602) is an atypical cannabinoid, potent and selective agonist of GPR55 cannabinoid receptor with EC50 of 13 nM, shows no significant activity for CB1 and CB2 receptors (EC50>30 uM). |
| PC-35195 |
ML193
GPR55 inhibitor
|
ML193 (CID 1261822) is a potent, selective GPR55 antagonist with IC50 of 221 nM, shows >27-, >145- and >145-fold selectivity for GPR55 over CB1, GPR35 and CB2, respectively. |
| PC-35027 |
ML191
GPR55 inhibitor
|
ML191 (CCG-152883) is a potent, selective GPR55 antagonist with 160 nM potency for GPR55 and >100-fold selectivity against GPR35, CB1 and CB2. |
| PC-35025 |
Abn-CBD
GPR55 agonist
|
Abn-CBD (Abnormal Cannabidiol) is a selective agonist of GPR55 receptor with EC50 of 2.5 uM, shows no significant activity against CB1 and CB2 receptors (EC50>30 uM). |
| PC-63115 |
GSK-575594A
GPR55 agonist
|
GSK-575594A is a potent, selective GPR55 agonist with pEC50 of 6.8 at GPR55 in yeast assay, displays 60-fold selective for GPR55 over GlyT1 (pIC50=5.0). |
| PC-70188 |
ML-184
GPR55 agonist
|
ML-184 (ML184) is a potent, selective GPR55 agonist with EC50 of 263 nM, >120-fold, 83-fold, and 57-fold selectivity against GPR35, CB1 and CB2. |
| PC-45043 |
CID16020046
GPR55 antagonist
|
CID16020046 is a potent and selective GPR55 antagonist with IC50 of 0.15 uM. |
| PC-21152 |
CID1792197
GPR55 agonist
|
CID1792197 is a potent, selective GPR55 agonist with EC50 of 110 nM in the β-arrestin trafficking assay,100-fold selectivity for GPR55 over GPR35, CB1 and CB2. |
