| Cat. No. |
Product Name |
Information |
| PC-38542 |
Takeda103A
GRK2 inhibitor
|
Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5. |
| PC-72421 |
GRK6 inhibitor 18
GRK6 inhibitor
|
GRK6 inhibitor 18 is a potent, and selective GRK6 inhibitor with IC50 of 8 nM. |
| PC-60588 |
CCG 258001
GRK2 inhibitor
|
CCG 258001 is a potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM. |
| PC-60587 |
CCG 224061
GRK2 inhibitor
|
A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM. |
| PC-60586 |
CCG 258748
GRK2 inhibitor
|
CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM. |
| PC-60585 |
Compound 101
GRK2/3 inhibitor
|
Compound 101 (GRK2 inhibitor 101, Takeda compound 101, Cmpd101) is a novel membrane-permeable, small-molecule inhibitor of GRK2 and GRK3 with IC50 of 18 nM and 5.4 nM, respectively. |
| PC-60353 |
GRK2-IN-115h hydrochloride
GRK2 inhibitor
|
GRK2-IN-115h hydrochloride is a highly potent and selective GRK2 inhibitor with IC50 of 18 nM. |
| PC-70119 |
CCG-224406
GRK2 inhibitor
|
CCG-224406 (CCG224406) is a highly selective and potent GRK2 (G protein-coupled receptor kinase 2) inhibitor with IC50 of 130 nM.M. |
| PC-45591 |
CCG215022
GRK inhibitor
|
CCG-215022 (CCG215022) is a potent and selective pan GRK (G protein-coupled receptor kinase) inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively. |
| PC-45590 |
GSK180736A
GRK2 inhibitor
|
GSK180736A is a highly selective and potent GRK2 inhibitor with IC50 of 0.77 uM. |
| PC-21461 |
GRL018-21
GRK5 inhibitor
|
GRL018-21 is a highly selective, potent, and non-covalent GRK5 inhibitor with IC50 of 10 nM, >100,000-fold selectivity over GRK2. |
