| Cat. No. |
Product Name |
Information |
| PC-61571 |
MCL0129 tetrahydrochloride
MC4R antagonist
|
MCL0129 tetrahydrochloride is a selective, potent melanocortin-4 receptor (MC4R) antagonist with Ki of 7.9 nM, without affinity for MC1 and MC3. |
| PC-61570 |
MCL0129
MC4R antagonist
|
MCL0129 is a selective, potent melanocortin-4 receptor (MC4R) antagonist with Ki of 7.9 nM, without affinity for MC1 and MC3. |
| PC-70138 |
Bremelanotide
Melanocortin receptor agonist
|
Bremelanotide (PT-141, PT141) is a peptide, non-selective melanocortin receptor agonist for treatment for female sexual dysfunction. |
| PC-60215 |
BMS-470539
MC-1R agonist
|
BMS-470539 is a potent, selective, full agonist of human and murine melanocortin-1 receptor (MC-1R) with EC50 of 16.8 and 11.6 nM, respectively. |
| PC-60214 |
PF-00446687
MC4R agonist
|
PF-00446687 (PF-446687) is a potent, selective melanocortin-4 receptor (MC4R) agonist with EC50 of 12 nM. |
| PC-60213 |
PF-00446687 hydrochloride
MC4R agonist
|
PF-00446687 hydrochloride (PF-446687) is a potent, selective melanocortin-4 receptor (MC4R) agonist with EC50 of 12 nM. |
| PC-70060 |
THIQ
MC4R agonist
|
THIQ is a potent and selective melanocortin 4 receptor (MC4R) agonist with EC50 of 2.1 nM. |
| PC-70059 |
SHU-9119
MC3R/MC4R antagonist
|
SHU-9119 is a potent melanocortin MC3 and MC4 receptor antagonist with IC50 of 0.23 nM and 0.06 nM, respectively. |
| PC-45520 |
Bremelanotide acetate
|
Bremelanotide acetate is an analogue of the naturally occurring peptide alpha-MSH. |
| PC-45743 |
Setmelanotide
Melanocortin receptor agonist
|
Setmelanotide (RM-493, BIM-22493, IRC-022493) is a peptide, non-selective melanocortin receptor agonist with binding Ki of 3.9/10/2.1 for hMC1R/hMC3R/hMC4R, respectively. |
| PC-49762 |
SNT-207707
MC4R inhibitor
|
SNT-207707 (SNT207707) is a potent, selective, BBB-penetrating, and orally active melanocortin-4 (MC-4) receptor antagonist with binding/fuaction IC50 of 8/5 nM, respectively. |
