| Cat. No. |
Product Name |
Information |
| PC-60266 |
CFI-401870
MPS1/TTK inhibitor
|
CFI-401870 is a potent, selective, orally active Mps1 (TTK) inhibitor with IC50 of 3.1 nM. |
| PC-60230 |
CCT271850
MPS1/TTK inhibitor
|
CCT271850 is a potent, selective, orally bioavailable Mps1 kinase (TTK) inhibitor with IC50 of 11 nM. |
| PC-42354 |
CFI-402257
MPS1/TTK inhibitor
|
CFI-402257 (CFI 402257) is a potent and selective Mps1/TTK kinase inhibitor with Ki of 0.1 nM and cellular Mps1 EC50 of 6.5 nM. |
| PC-22996 |
BAL0891
TTK/PLK1 inhibitor
|
BAL0891 is a first in class, potent dual TTK/PLK1 inhibitor with IC50 of 0.4/46 nM respectively. |
| PC-22995 |
AZ3146
Mps1 inhibitor
|
AZ3146 is a potent selective Mps1 inhibitor with IC50 of 35 nM against human Mps1Cat. |
| PC-21597 |
SYL1073
MPS1/TTK inhibitor
|
SYL1073 is a potent, selective and covalent Threonine tyrosine kinase (TTK) inhibitor with IC50 of of 16 nM. |
| PC-21558 |
PF-3837
MPS1/TTK inhibitor
|
PF-3837 is a potent, highly-selective Mps1 (TTK) inhibitor with Ki of 0.33 nM, potently inhibit Mps1 in MDA-MB-468 tumor cells with IC50 of 5.5 nM. |
| PC-21557 |
PF-7006
MPS1/TTK inhibitor
|
PF-7006 is a potent, highly-selective Mps1 (TTK) inhibitor with Ki of 0.27 nM, potently inhibit Mps1 in MDA-MB-468 tumor cells with IC50 of 2.5 nM. |
| PC-21556 |
CFI-400936
MPS1/TTK inhibitor
|
CFI-400936 is a potent, selective Tyrosine Threonine Kinase (TTK, Mps1) inhibitor with IC50 of 3.6 nM. |
